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Lead Optimization: The synthetic modification of a biologically active compound, to fulfill all stereoelectronic, physicochemical, pharmacokinetic and toxicologic required for clinical usefulness.

Contract Pharmaceutical/Lead Optimization Research Services that can be outsourced on CanBiotech include:

Chemistry
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  Combinatorial Chemistry/Library Development
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  Organic Chemical Synthesis

Drug Development
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  Efficacy Studies
  Formulation
  Screening
  Synthesis
  Toxicology Studies

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